收录：
摘要：
A series of novel 6-(pyrazolylmethyl)-4-oxo-4H-quinoline-3-carboxylic acid derivatives bearing different substituents on the N-position of quinoline ring were designed and synthesized as potential HIV-1 integrase (IN) inhibitors, based on the structurally related GS-9137 scaffold. The structures of all new compounds were confirmed by H-1-NMR, C-13-NMR and ESI (or HRMS) spectra. Detailed synthetic protocols and the anti-IN activity studies are also presented.
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电子邮件地址：
来源 ：
MOLECULES
ISSN： 1420-3049
年份： 2012
期： 9
卷： 17
页码： 10652-10666
4 . 6 0 0
JCR@2022
ESI学科： CHEMISTRY;
JCR分区：2
中科院分区：3
